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Assay Detail

CHEMBL747315

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity of compound against human normal neonatal foreskin fibroblasts (NFF) cell line
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type NFF
Confidence 1 — Organism
Curated By Intermediate

Target

NFF (CHEMBL614198)
Type CELL-LINE
Organism Homo sapiens

Publication

Antiproliferative and phenotype-transforming antitumor agents derived from cysteine.
Glenn MP, Kahnberg P, Boyle GM, Hansford KA, Hans D, Martyn AC, Parsons PG, Fairlie DP.
J Med Chem (2004) 47 : 2984 -2994
PubMed 15163181 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.19 6.46

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL318384 1 6.46
CHEMBL101006 1 6.10
CHEMBL103508 1 6.10
CHEMBL103379 1 6.08

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL318384 IC50 = 350.0 nM 6.46
CHEMBL101006 IC50 = 800.0 nM 6.10
CHEMBL103508 IC50 = 800.0 nM 6.10
CHEMBL103379 IC50 = 830.0 nM 6.08