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Assay Detail

CHEMBL748858

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards nicotinic acetylcholine receptor using [125I]alpha-bungarotoxin as radioligand in rat forebrain homogenates
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Tissue Brain
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Neuronal acetylcholine receptor (CHEMBL2094110)
Type PROTEIN COMPLEX GROUP
Organism Rattus norvegicus

Publication

Rigidified acetylcholine mimics: conformational requirements for binding to neuronal nicotinic receptors.
Villeneuve G, Cécyre D, Lejeune H, Drouin M, Lan R, Quirion R.
Bioorg Med Chem Lett (2003) 13 : 3847 -3851
PubMed 14552793 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 34 5.42 8.43

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL6623 EPIBATIDINE 1 8.43
CHEMBL25619 1 8.40
CHEMBL338918 1 6.82
CHEMBL338558 1 6.80
CHEMBL124471 1 6.77
CHEMBL125190 1 6.68
CHEMBL338316 1 5.62
CHEMBL609401 1 5.57
CHEMBL609144 1 5.55
CHEMBL126222 1 5.54
CHEMBL420150 1 5.27
CHEMBL126015 1 4.91
CHEMBL609140 1 4.82
CHEMBL122270 LOBELINE 2.0 1 4.74
CHEMBL435616 1 4.60
CHEMBL609406 1 4.51
CHEMBL609146 1 4.43
CHEMBL332008 1 4.37
CHEMBL609145 1 4.36
CHEMBL612094 1 4.30
CHEMBL612097 1 4.09
CHEMBL126527 1 4.06
CHEMBL127640 1 4.04
CHEMBL332009 1 -
CHEMBL126637 1 -
CHEMBL612093 1 -
CHEMBL340079 1 -
CHEMBL1161006 1 -
CHEMBL609142 1 -
CHEMBL339474 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL6623 EPIBATIDINE IC50 = 3.7 nM 8.43
CHEMBL25619 IC50 = 4.0 nM 8.40
CHEMBL338918 IC50 = 150.0 nM 6.82
CHEMBL338558 IC50 = 160.0 nM 6.80
CHEMBL124471 IC50 = 170.0 nM 6.77
CHEMBL125190 IC50 = 210.0 nM 6.68
CHEMBL338316 IC50 = 2400.0 nM 5.62
CHEMBL609401 IC50 = 2720.0 nM 5.57
CHEMBL609144 IC50 = 2800.0 nM 5.55
CHEMBL126222 IC50 = 2870.0 nM 5.54
CHEMBL420150 IC50 = 5400.0 nM 5.27
CHEMBL126015 IC50 = 12200.0 nM 4.91
CHEMBL609140 IC50 = 15000.0 nM 4.82
CHEMBL122270 LOBELINE IC50 = 18100.0 nM 4.74
CHEMBL435616 IC50 = 25300.0 nM 4.60
CHEMBL609406 IC50 = 31000.0 nM 4.51
CHEMBL609146 IC50 = 37000.0 nM 4.43
CHEMBL332008 IC50 = 43000.0 nM 4.37
CHEMBL609145 IC50 = 44000.0 nM 4.36
CHEMBL612094 IC50 = 49500.0 nM 4.30
CHEMBL612097 IC50 = 81000.0 nM 4.09
CHEMBL126527 IC50 = 87000.0 nM 4.06
CHEMBL127640 IC50 = 91000.0 nM 4.04
CHEMBL332009 IC50 = 207000.0 nM -
CHEMBL126637 IC50 > 100000.0 nM -
CHEMBL612093 IC50 = 111000.0 nM -
CHEMBL340079 IC50 > 100000.0 nM -
CHEMBL1161006 IC50 > 100000.0 nM -
CHEMBL609142 IC50 > 100000.0 nM -
CHEMBL339474 IC50 = 134000.0 nM -
CHEMBL609404 IC50 > 100000.0 nM -
CHEMBL609399 IC50 = 115000.0 nM -
CHEMBL609402 IC50 > 100000.0 nM -
CHEMBL1161007 IC50 = 436000.0 nM -