Assay Detail
Functional
CHEMBL749398
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of phorbol-12-myristate-13-acetate (PMA)induced superoxide burst in human neutrophils
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Synthesis and protein kinase inhibitory activity of balanol analogues with modified benzophenone subunits.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 5.44 | 6.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL91126 | — | — | 1 | 6.33 |
| CHEMBL89639 | — | — | 1 | 5.82 |
| CHEMBL328747 | — | — | 1 | 5.04 |
| CHEMBL88749 | — | — | 1 | 5.00 |
| CHEMBL89591 | — | — | 1 | 5.00 |
| CHEMBL312846 | — | — | 1 | - |
| CHEMBL89384 | — | — | 1 | - |
| CHEMBL89648 | — | — | 1 | - |
| CHEMBL421539 | — | — | 1 | - |
| CHEMBL433361 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL91126 | — | IC50 | = | 470.0 | nM | 6.33 |
| CHEMBL89639 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL328747 | — | IC50 | = | 9200.0 | nM | 5.04 |
| CHEMBL88749 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL89591 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL312846 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL89384 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL89648 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL421539 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL433361 | — | IC50 | > | 10000.0 | nM | - |