Assay Detail
Functional
CHEMBL750156
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Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of human erythrocytes
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Purine and pyrimidine (P2) receptors as drug targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 6.00 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL69234 | — | — | 1 | 6.00 |
| CHEMBL336296 | URIDINE TRIPHOSPHATE | 3.0 | 1 | - |
| CHEMBL130266 | URIDINE_DIPHOSPHATE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL69234 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL336296 | URIDINE TRIPHOSPHATE | EC50 | > | 100000.0 | nM | - |
| CHEMBL130266 | URIDINE_DIPHOSPHATE | EC50 | > | 100000.0 | nM | - |