Assay Detail
Binding
CHEMBL751074
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity against Opioid receptor mu 1 with [3H]CTOP
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Topographical requirements for delta opioid ligands: The synthesis and biological properties of a cyclic analogue of deltorphin I
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.98 | 8.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL153466 | — | — | 1 | 8.29 |
| CHEMBL317956 | DELTORPHIN C | — | 1 | 5.67 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL153466 | — | IC50 | = | 5.15 | nM | 8.29 |
| CHEMBL317956 | DELTORPHIN C | IC50 | = | 2140.0 | nM | 5.67 |