Assay Detail
Functional
CHEMBL751483
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Selective inhibition of serum stimulated growth of NIH3T3neu isogenic cells
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | NIH3T3 |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
The combi-targeting concept: chemical dissection of the dual targeting properties of a series of "combi-triazenes".
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 4.99 | 5.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL137364 | — | — | 1 | 5.54 |
| CHEMBL136674 | — | — | 1 | 5.53 |
| CHEMBL136491 | — | — | 1 | 5.51 |
| CHEMBL137534 | — | — | 1 | 5.47 |
| CHEMBL134312 | — | — | 1 | 5.43 |
| CHEMBL138125 | — | — | 1 | 5.39 |
| CHEMBL52765 | — | — | 1 | 5.39 |
| CHEMBL133024 | — | — | 1 | 5.38 |
| CHEMBL137617 | — | — | 1 | 5.37 |
| CHEMBL343352 | — | — | 1 | 5.31 |
| CHEMBL133023 | — | — | 1 | 5.16 |
| CHEMBL336113 | — | — | 1 | 5.14 |
| CHEMBL137189 | — | — | 1 | 5.01 |
| CHEMBL424093 | — | — | 1 | 4.95 |
| CHEMBL344652 | — | — | 1 | 4.50 |
| CHEMBL332096 | — | — | 1 | 4.47 |
| CHEMBL137027 | — | — | 1 | 4.47 |
| CHEMBL137788 | — | — | 1 | 4.46 |
| CHEMBL137635 | — | — | 1 | 4.19 |
| CHEMBL135592 | — | — | 1 | 4.09 |
| CHEMBL136492 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL137364 | — | IC50 | = | 2920.0 | nM | 5.54 |
| CHEMBL136674 | — | IC50 | = | 2980.0 | nM | 5.53 |
| CHEMBL136491 | — | IC50 | = | 3090.0 | nM | 5.51 |
| CHEMBL137534 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL134312 | — | IC50 | = | 3740.0 | nM | 5.43 |
| CHEMBL138125 | — | IC50 | = | 4060.0 | nM | 5.39 |
| CHEMBL52765 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL133024 | — | IC50 | = | 4160.0 | nM | 5.38 |
| CHEMBL137617 | — | IC50 | = | 4320.0 | nM | 5.37 |
| CHEMBL343352 | — | IC50 | = | 4930.0 | nM | 5.31 |
| CHEMBL133023 | — | IC50 | = | 6940.0 | nM | 5.16 |
| CHEMBL336113 | — | IC50 | = | 7200.0 | nM | 5.14 |
| CHEMBL137189 | — | IC50 | = | 9690.0 | nM | 5.01 |
| CHEMBL424093 | — | IC50 | = | 11230.0 | nM | 4.95 |
| CHEMBL344652 | — | IC50 | = | 31640.0 | nM | 4.50 |
| CHEMBL332096 | — | IC50 | = | 33790.0 | nM | 4.47 |
| CHEMBL137027 | — | IC50 | = | 33900.0 | nM | 4.47 |
| CHEMBL137788 | — | IC50 | = | 34910.0 | nM | 4.46 |
| CHEMBL137635 | — | IC50 | = | 64090.0 | nM | 4.19 |
| CHEMBL135592 | — | IC50 | = | 81050.0 | nM | 4.09 |
| CHEMBL136492 | — | IC50 | = | 99370.0 | nM | 4.00 |