Assay Detail
Binding
CHEMBL752035
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against Opioid receptor mu 1 of (endomorphin 2) in guinea pig ileum was determined
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Tissue | Ileum |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Enkephalin analogues with 2',6'-dimethylphenylalanine replacing phenylalanine in position 4.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.90 | 6.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL111028 | — | — | 1 | 6.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL111028 | — | Kd | = | 125.89 | nM | 6.90 |