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Assay Detail

CHEMBL754113

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Binding
Binding affinity to nucleotide-binding domain (NBD2) of P-Glycoprotein
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

ATP-dependent translocase ABCB1 (CHEMBL2573)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

B-ring substituted 5,7-dihydroxyflavonols with high-affinity binding to P-glycoprotein responsible for cell multidrug resistance.
Boumendjel A, Bois F, Beney C, Mariotte AM, Conseil G, Di Pietro A.
Bioorg Med Chem Lett (2001) 11 : 75 -77
PubMed 11140738 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 8 5.65 7.24

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL164611 1 7.24
CHEMBL166368 1 5.97
CHEMBL164555 1 5.70
CHEMBL165607 1 5.40
CHEMBL40919 KAEMPFERIDE 1 5.30
CHEMBL309490 GALANGIN 1 5.23
CHEMBL150 KAEMPFEROL 1.0 1 5.17
CHEMBL165905 1 5.17

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL164611 Kd = 57.0 nM 7.24
CHEMBL166368 Kd = 1060.0 nM 5.97
CHEMBL164555 Kd = 2000.0 nM 5.70
CHEMBL165607 Kd = 4000.0 nM 5.40
CHEMBL40919 KAEMPFERIDE Kd = 5000.0 nM 5.30
CHEMBL309490 GALANGIN Kd = 5900.0 nM 5.23
CHEMBL150 KAEMPFEROL Kd = 6700.0 nM 5.17
CHEMBL165905 Kd = 6800.0 nM 5.17