Assay Detail
Binding
CHEMBL754143
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Opioid receptor activity was evaluated using mouse vas deferens (MVD) assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Tissue | Vas deferens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.58 | 8.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1790710 | — | — | 1 | 8.57 |
| CHEMBL70 | MORPHINE | 4.0 | 1 | 6.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1790710 | — | IC50 | = | 2.7 | nM | 8.57 |
| CHEMBL70 | MORPHINE | IC50 | = | 258.0 | nM | 6.59 |