Assay Detail
Binding
CHEMBL754348
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Equilibrium dissociation constant at cloned rat Neurotensin receptor (NT) receptor expressed in CHO-K1 cells; 0.3-0.7 uM
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | CHO-K1 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Synthesis of partially non-peptidic neurotensin mimetics
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 6.52 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL21521 | — | — | 1 | 6.52 |
| CHEMBL21448 | — | — | 1 | 6.52 |
| CHEMBL21892 | — | — | 1 | 6.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL21521 | — | Kd | = | 300.0 | nM | 6.52 |
| CHEMBL21448 | — | Kd | = | 300.0 | nM | 6.52 |
| CHEMBL21892 | — | Kd | = | 300.0 | nM | 6.52 |