Assay Detail
Functional
CHEMBL754797
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The compound was tested for competitive antagonist of Nitric oxide synthase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Examination of N-hydroxylation as a prerequisite mechanism of nitric oxide synthase inactivation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 4.83 | 5.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL7889 | L-NIL | — | 1 | 5.67 |
| CHEMBL269180 | — | — | 1 | 4.42 |
| CHEMBL556931 | — | — | 1 | 4.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL7889 | L-NIL | Ki | = | 2160.0 | nM | 5.67 |
| CHEMBL269180 | — | Ki | = | 37700.0 | nM | 4.42 |
| CHEMBL556931 | — | Ki | = | 41100.0 | nM | 4.39 |