Assay Detail
Binding
CHEMBL756766
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Binding affinity for porcine Pancreatic elastase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Chymotrypsin-like elastase family member 2A (CHEMBL2407) ↗| Type | SINGLE PROTEIN |
| Organism | Sus scrofa |
Publication
Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.30 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL79463 | — | — | 1 | 7.89 |
| CHEMBL55210 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL79463 | — | Ki | = | 13.0 | nM | 7.89 |
| CHEMBL55210 | — | Ki | = | 200.0 | nM | 6.70 |