Assay Detail
Binding
CHEMBL756767
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards porcine pancreatic elastase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Chymotrypsin-like elastase family member 2A (CHEMBL2407) ↗| Type | SINGLE PROTEIN |
| Organism | Sus scrofa |
Publication
Peptidyl alpha-ketoheterocyclic inhibitors of human neutrophil elastase. 3. In vitro and in vivo potency of a series of peptidyl alpha-ketobenzoxazoles.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.58 | 7.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL419985 | — | — | 1 | 7.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL419985 | — | Ki | = | 26.0 | nM | 7.58 |