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Assay Detail

CHEMBL756822

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibitory activity against IgE antibody production in PBMC
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

ADMET (CHEMBL612558)
Type ADMET

Publication

Novel naphthalene derivatives as inhibitors of human immunoglobulin E antibody production.
Hasegawa M, Takenouchi K, Takahashi K, Takeuchi T, Komoriya K, Uejima Y, Kamimura T.
J Med Chem (1997) 40 : 395 -407
PubMed 9046329 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.82 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL336392 1 5.92
CHEMBL337497 1 5.80
CHEMBL133470 1 5.73

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL336392 IC50 = 1200.0 nM 5.92
CHEMBL337497 IC50 = 1570.0 nM 5.80
CHEMBL133470 IC50 = 1880.0 nM 5.73