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Assay Detail

CHEMBL757537

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards Opioid receptor delta 1
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Delta-type opioid receptor (CHEMBL3222)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Solid phase synthesis and evaluation of Tyr-Tic-Phe-Phe(p-NHCOCH(2)Br) ([Phe(p-bromoacetamide)(4)]TIPP), a potent affinity label for delta opioid receptors.
Kumar V, Murray TF, Aldrich JV.
J Med Chem (2002) 45 : 3820 -3823
PubMed 12190304 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.91 8.91

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL191751 1 8.91

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL191751 Ki = 1.22 nM 8.91