Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL757783

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards peroxisome proliferator activated receptor alpha (murinePPAR alpha)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Peroxisome proliferator-activated receptor alpha (CHEMBL2128)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

O-arylmandelic acids as highly selective human PPAR alpha/gamma agonists.
Adams AD, Hu Z, von Langen D, Dadiz A, Elbrecht A, MacNaul KL, Berger JP, Zhou G, Doebber TW, Meurer R, Forrest MJ, Moller DE, Jones AB.
Bioorg Med Chem Lett (2003) 13 : 3185 -3190
PubMed 12951090 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.00 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL295416 PIRINIXIC ACID 2.0 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL295416 PIRINIXIC ACID Ki = 100.0 nM 7.00