Assay Detail
Binding
CHEMBL757996
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against delta receptor of (endomorphin 2) in mouse vas deferens was determined
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Vas deferens |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Enkephalin analogues with 2',6'-dimethylphenylalanine replacing phenylalanine in position 4.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 5.59 | 5.59 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL111028 | — | — | 1 | 5.59 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL111028 | — | Kd | = | 2570.4 | nM | 5.59 |