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Assay Detail

CHEMBL758001

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Negative logarithm of the molar concentration of delta receptor was determined in mouse vas deferens
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Delta-type opioid receptor (CHEMBL3222)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Assessment of substitution in the second pharmacophore of Dmt-Tic analogues.
Santagada V, Balboni G, Caliendo G, Guerrini R, Salvadori S, Bianchi C, Bryant SD, Lazarus LH.
Bioorg Med Chem Lett (2000) 10 : 2745 -2748
PubMed 11133082 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 9.48 9.48

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL296603 DELTORPHINE II 1 9.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL296603 DELTORPHINE II EC50 = 0.3311 nM 9.48