Assay Detail
Functional
CHEMBL759541
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was tested for displacement of 3[H] oxytocin from rat OT receptor (in vitro)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of potent and selective oxytocin antagonists. Part 2: further investigation of benzofuran derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.19 | 6.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL24781 | — | — | 1 | 6.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL24781 | — | IC50 | = | 640.0 | nM | 6.19 |