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Assay Detail

CHEMBL760372

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of [3H]- PDBu binding to peptide C, rat brain PKC gamma
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Protein kinase C gamma type (CHEMBL3604)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Synthesis and characterization of the second cysteine-rich region of mouse skin PKCGh
Irie K, Yanai Y, Ohigashi H, Wender PA, Miller BL
Bioorg Med Chem Lett (1996) 6 : 353 -356
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.70 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL417692 1 8.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL417692 Ki = 2.0 nM 8.70