Assay Detail
Binding
CHEMBL761407
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The inhibition constant (Ki(nM)) by displacement of [125I]- HO-LVA radiolabeled ligand using membranes of CHO cells of human Oxytocin receptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Fluorescent pseudo-peptide linear vasopressin antagonists: design, synthesis, and applications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 8.81 | 8.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL262035 | — | — | 1 | 8.96 |
| CHEMBL540192 | — | — | 1 | 8.92 |
| CHEMBL412210 | — | — | 1 | 8.80 |
| CHEMBL269012 | — | — | 1 | 8.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL262035 | — | Ki | = | 1.1 | nM | 8.96 |
| CHEMBL540192 | — | Ki | = | 1.2 | nM | 8.92 |
| CHEMBL412210 | — | Ki | = | 1.6 | nM | 8.80 |
| CHEMBL269012 | — | Ki | = | 2.7 | nM | 8.57 |