Assay Detail
Binding
CHEMBL765785
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Compound was evaluated for binding inhibition against Prolyl Endopeptidase (PEP).
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Novel in vitro and in vivo inhibitors of prolyl endopeptidase
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.55 | 8.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL345903 | — | — | 1 | 8.62 |
| CHEMBL154968 | — | — | 1 | 8.52 |
| CHEMBL155614 | — | — | 1 | 8.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL345903 | — | Ki | = | 2.4 | nM | 8.62 |
| CHEMBL154968 | — | Ki | = | 3.0 | nM | 8.52 |
| CHEMBL155614 | — | Ki | = | 3.0 | nM | 8.52 |