Assay Detail
Binding
CHEMBL766948
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was tested for inhibitory activity against prostaglandin synthetase in mouse brain microsomes
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Brain |
| Subcellular | Microsome |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Morpholinoalkylindenes as antinociceptive agents: Novel cannabinoid receptor agonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.08 | 5.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL13178 | PRAVADOLINE | 2.0 | 1 | 5.46 |
| CHEMBL129525 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL13178 | PRAVADOLINE | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL129525 | — | IC50 | = | 20000.0 | nM | 4.70 |