Assay Detail
Binding
CHEMBL767033
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Inhibition of Protein kinase C alpha
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Kinase inhibitors: not just for kinases anymore.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.59 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL268769 | — | — | 1 | 7.70 |
| CHEMBL6291 | BISINDOLYLMALEIMIDE IX | — | 1 | 7.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL268769 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL6291 | BISINDOLYLMALEIMIDE IX | IC50 | = | 33.0 | nM | 7.48 |