Assay Detail
Binding
CHEMBL767398
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C eta
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis and characterization of the second cysteine-rich region of mouse skin PKCGh
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 8.88 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL417692 | — | — | 1 | 10.00 |
| CHEMBL27768 | — | — | 1 | 9.22 |
| CHEMBL120645 | — | — | 1 | 8.47 |
| CHEMBL24609 | MONOCTANOIN COMPONENT C | -1.0 | 1 | 7.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL417692 | — | Ki | = | 0.1 | nM | 10.00 |
| CHEMBL27768 | — | Ki | = | 0.6 | nM | 9.22 |
| CHEMBL120645 | — | Ki | = | 3.36 | nM | 8.47 |
| CHEMBL24609 | MONOCTANOIN COMPONENT C | Ki | = | 14.5 | nM | 7.84 |