Assay Detail
Binding
CHEMBL767405
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]- PDBu from Protein kinase C eta C1a domain
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Synthesis and PKC isozyme surrogate binding of indothiolactam-V, a new thioamide analogue of tumor promoting indolactam-V.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.55 | 5.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL63262 | — | — | 1 | 5.67 |
| CHEMBL27266 | INDOLACTUM | — | 1 | 5.42 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL63262 | — | Ki | = | 2160.0 | nM | 5.67 |
| CHEMBL27266 | INDOLACTUM | Ki | = | 3770.0 | nM | 5.42 |