Assay Detail
Binding
CHEMBL767784
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The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of LAR
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Tyrosine-protein phosphatase non-receptor type 1 (CHEMBL335) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Synthesis and characterization of a potent and selective protein tyrosine phosphatase inhibitor, 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.63 | 4.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL89067 | — | — | 1 | 4.74 |
| CHEMBL86473 | VANADATE | — | 1 | 4.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL89067 | — | IC50 | = | 18200.0 | nM | 4.74 |
| CHEMBL86473 | VANADATE | IC50 | = | 30800.0 | nM | 4.51 |