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Assay Detail

CHEMBL768750

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
In vitro inhibitory activity against human whole blood Prostaglandin G/H synthase 1
9
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Prostaglandin G/H synthase 1 (CHEMBL221)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

The discovery of rofecoxib, [MK 966, Vioxx, 4-(4'-methylsulfonylphenyl)-3-phenyl-2(5H)-furanone], an orally active cyclooxygenase-2-inhibitor.
Prasit P, Wang Z, Brideau C, Chan CC, Charleson S, Cromlish W, Ethier D, Evans JF, Ford-Hutchinson AW, Gauthier JY, Gordon R, Guay J, Gresser M, Kargman S, Kennedy B, Leblanc Y, Léger S, Mancini J, O'Neill GP, Ouellet M, Percival MD, Perrier H, Riendeau D, Rodger I, Zamboni R.
Bioorg Med Chem Lett (1999) 9 : 1773 -1778
PubMed 10406640 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 9 5.26 6.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL139 DICLOFENAC 4.0 1 6.82
CHEMBL6 INDOMETHACIN 4.0 1 6.70
CHEMBL431546 1 5.24
CHEMBL118 CELECOXIB 4.0 1 5.20
CHEMBL51434 1 5.00
CHEMBL18264 1 4.89
CHEMBL122 ROFECOXIB 4.0 2 4.72
CHEMBL52285 1 4.07

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL139 DICLOFENAC IC50 = 150.0 nM 6.82
CHEMBL6 INDOMETHACIN IC50 = 200.0 nM 6.70
CHEMBL431546 IC50 = 5800.0 nM 5.24
CHEMBL118 CELECOXIB IC50 = 6300.0 nM 5.20
CHEMBL51434 IC50 = 10000.0 nM 5.00
CHEMBL18264 IC50 = 13000.0 nM 4.89
CHEMBL122 ROFECOXIB IC50 = 19000.0 nM 4.72
CHEMBL122 ROFECOXIB IC50 = 19000.0 nM 4.72
CHEMBL52285 IC50 = 86000.0 nM 4.07