Assay Detail
Functional
CHEMBL779561
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro inhibitory concentration for 50% relaxant effect was measured on rat bladder strips
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Recent developments in the biology and medicinal chemistry of potassium channel modulators: update from a decade of progress.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.03 | 7.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2062142 | — | — | 1 | 7.05 |
| CHEMBL2062143 | — | — | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2062142 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL2062143 | — | IC50 | = | 100.0 | nM | 7.00 |