Assay Detail
Functional
CHEMBL782135
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against graft vs host disease in rat.
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Selective inhibitors of protein kinase C in a model of graft-vs-host disease
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.31 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL79682 | — | — | 1 | 5.80 |
| CHEMBL80111 | — | — | 1 | 5.60 |
| CHEMBL311192 | — | — | 1 | 5.58 |
| CHEMBL80658 | — | — | 1 | 5.54 |
| CHEMBL80059 | — | — | 1 | 5.52 |
| CHEMBL79836 | — | — | 1 | 5.52 |
| CHEMBL79798 | — | — | 1 | 5.47 |
| CHEMBL80058 | — | — | 1 | 5.44 |
| CHEMBL309772 | — | — | 1 | 5.43 |
| CHEMBL82547 | — | — | 1 | 5.38 |
| CHEMBL78466 | — | — | 1 | 5.38 |
| CHEMBL309386 | — | — | 1 | 5.36 |
| CHEMBL431593 | — | — | 1 | 5.35 |
| CHEMBL83332 | — | — | 1 | 5.32 |
| CHEMBL311475 | — | — | 1 | 5.24 |
| CHEMBL431004 | — | — | 1 | 5.24 |
| CHEMBL313402 | — | — | 1 | 5.21 |
| CHEMBL311068 | — | — | 1 | 5.15 |
| CHEMBL309437 | — | — | 1 | 5.10 |
| CHEMBL81130 | — | — | 1 | 4.96 |
| CHEMBL314696 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL79682 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL80111 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL311192 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL80658 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL80059 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL79836 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL79798 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL80058 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL309772 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL82547 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL78466 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL309386 | — | IC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL431593 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL83332 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL311475 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL431004 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL313402 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL311068 | — | IC50 | = | 7100.0 | nM | 5.15 |
| CHEMBL309437 | — | IC50 | = | 7900.0 | nM | 5.10 |
| CHEMBL81130 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL314696 | — | IC50 | = | 100000.0 | nM | 4.00 |