Assay Detail
Functional
CHEMBL782322
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Compound was tested for inhibition of glucose transport in adipocytes plasma membrane vesicles using [H]-forskolin as radioligand
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
On the analogy between forskolin and D-glucose.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.89 | 6.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL52606 | COLFORSIN | 2.0 | 1 | 6.62 |
| CHEMBL486619 | — | — | 1 | 5.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL52606 | COLFORSIN | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL486619 | — | EC50 | = | 7100.0 | nM | 5.15 |