Assay Detail
Functional
CHEMBL783635
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Antagonist activity against amylase secretion from rat pancreatic acini
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
On the significance of the C-terminal primary amide in cholecystokinin
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.55 | 4.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL413186 | — | — | 1 | 4.58 |
| CHEMBL216527 | — | — | 1 | 4.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL413186 | — | IC50 | = | 26000.0 | nM | 4.58 |
| CHEMBL216527 | — | IC50 | = | 30000.0 | nM | 4.52 |