Assay Detail
Functional
CHEMBL797693
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory concentration for [3H]PCP binding to rat brain homogenate relative to PCP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Tissue | Brain |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Structure-activity relationships of the cycloalkyl ring of phencyclidine.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.57 | 6.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL542581 | PHENCYCLIDINE HYDROCHLORIDE | -1.0 | 1 | 6.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL542581 | PHENCYCLIDINE HYDROCHLORIDE | IC50 | = | 270.0 | nM | 6.57 |