Assay Detail
Functional
CHEMBL798755
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Electropharmacology on rat cortical slice preparation for EAA-evoked depolarizations;Depolarization evoked by the compound is partially antagonised by 5 uM of NBQX and fully antagonised by 20 uM of NBQX.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.46 | 5.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL125440 | — | — | 1 | 5.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL125440 | — | EC50 | = | 3500.0 | nM | 5.46 |