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Assay Detail

CHEMBL800380

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was evaluated for its inhibitory concentration against [Fe2+]/AA- induced oxidative neuronal damage in primary cultured rat cortical cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Confidence 1 — Organism
Curated By Intermediate

Target

Rattus norvegicus (CHEMBL376)
Type ORGANISM
Organism Rattus norvegicus

Publication

Synthesis and evaluation of 4-hydroxyphenylacetic acid amides and 4-hydroxycinnamamides as antioxidants.
Jung YS, Kang TS, Yoon JH, Joe BY, Lim HJ, Seong CM, Park WK, Kong JY, Cho J, Park NS.
Bioorg Med Chem Lett (2002) 12 : 2599 -2602
PubMed 12182869 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.94 5.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL87037 1 5.62
CHEMBL312901 1 4.62
CHEMBL86670 1 4.57
CHEMBL153 TROLOX 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL87037 IC50 = 2400.0 nM 5.62
CHEMBL312901 IC50 = 23700.0 nM 4.62
CHEMBL86670 IC50 = 26800.0 nM 4.57
CHEMBL153 TROLOX IC50 = 430530.0 nM -