Assay Detail
Functional
CHEMBL802703
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was evaluated for the inhibition of insulin release from rat islets
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Rattus norvegicus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Phenylcyanoguanidines as inhibitors of glucose-induced insulin secretion from beta cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.21 | 5.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL181 | DIAZOXIDE | 4.0 | 1 | 5.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL181 | DIAZOXIDE | IC50 | = | 6100.0 | nM | 5.21 |