Assay Detail
Binding
CHEMBL803857
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Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR4
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 9.31 | 10.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1823872 | SOMATOSTATIN | 3.0 | 1 | 10.10 |
| CHEMBL3350037 | — | — | 1 | 8.52 |
| CHEMBL306702 | — | — | 1 | - |
| CHEMBL421493 | — | — | 1 | - |
| CHEMBL266469 | — | — | 1 | - |
| CHEMBL69379 | — | — | 1 | - |
| CHEMBL436783 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1823872 | SOMATOSTATIN | IC50 | = | 0.08 | nM | 10.10 |
| CHEMBL3350037 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL306702 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL421493 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL266469 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL69379 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL436783 | — | IC50 | > | 1000.0 | nM | - |