Assay Detail
Binding
CHEMBL804767
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity of compound against SSAT extracted from superinduced H157 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | H157 |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Terminally alkylated polyamine analogues as chemotherapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.20 | 4.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL86940 | — | — | 1 | 4.40 |
| CHEMBL33387 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL86940 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL33387 | — | IC50 | = | 100000.0 | nM | 4.00 |