Assay Detail
Binding
CHEMBL806596
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Tested for inhibition of radioligand binding to cloned somatostatin receptor hSSTR5
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 8.44 | 9.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3350037 | — | — | 1 | 9.11 |
| CHEMBL266469 | — | — | 1 | 8.38 |
| CHEMBL436783 | — | — | 1 | 8.31 |
| CHEMBL421493 | — | — | 1 | 7.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3350037 | — | IC50 | = | 0.77 | nM | 9.11 |
| CHEMBL266469 | — | IC50 | = | 4.17 | nM | 8.38 |
| CHEMBL436783 | — | IC50 | = | 4.92 | nM | 8.31 |
| CHEMBL421493 | — | IC50 | = | 10.95 | nM | 7.96 |