Assay Detail
Binding
CHEMBL806602
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Compound was tested for the inhibition of rSSTR5
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A refined model for the somatostatin pharmacophore: conformational analysis of lanthionine-sandostatin analogs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 8.08 | 8.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL415860 | — | — | 1 | 8.98 |
| CHEMBL266469 | — | — | 1 | 8.89 |
| CHEMBL436783 | — | — | 1 | 8.26 |
| CHEMBL421493 | — | — | 1 | 7.97 |
| CHEMBL69379 | — | — | 1 | 6.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL415860 | — | IC50 | = | 1.04 | nM | 8.98 |
| CHEMBL266469 | — | IC50 | = | 1.29 | nM | 8.89 |
| CHEMBL436783 | — | IC50 | = | 5.5 | nM | 8.26 |
| CHEMBL421493 | — | IC50 | = | 10.63 | nM | 7.97 |
| CHEMBL69379 | — | IC50 | = | 500.0 | nM | 6.30 |