Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL806839

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was tested for the inhibition of spinal reflex evoked by electrical stimulation of the dorsal root of new born rat
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Confidence 1 — Organism
Curated By Intermediate

Target

Rattus norvegicus (CHEMBL376)
Type ORGANISM
Organism Rattus norvegicus

Publication

Syntheses and conformational analyses of glutamate analogs: 2-(2-carboxy-3-substituted-cyclopropyl)glycines as useful probes for excitatory amino acid receptors.
Shimamoto K, Ohfune Y.
J Med Chem (1996) 39 : 407 -423
PubMed 8558509 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.16 6.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL280563 1 6.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL280563 IC50 = 700.0 nM 6.16