Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL807654

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity on rat 5-alpha reductase-2 isozyme
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

3-oxo-5-alpha-steroid 4-dehydrogenase 2 (CHEMBL5099)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Pharmacological options in the treatment of benign prostatic hyperplasia.
Kenny B, Ballard S, Blagg J, Fox D.
J Med Chem (1997) 40 : 1293 -1315
PubMed 9135028 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL24955 BEXLOSTERIDE 2.0 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL24955 BEXLOSTERIDE Ki = 10000.0 nM 5.00