Assay Detail
Functional
CHEMBL810908
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonistic activity as progesterone receptor induced alkaline phosphatase activity in T47D human breast cancer cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T47D |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Novel pyrrole-containing progesterone receptor modulators.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.85 | 8.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL67860 | — | — | 1 | 8.96 |
| CHEMBL431380 | — | — | 1 | 8.74 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL67860 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL431380 | — | EC50 | = | 1.8 | nM | 8.74 |