Assay Detail
Binding
CHEMBL813871
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Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligand
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
The design of polar -turn dipeptide mimetics
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 5.35 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL33650 | — | — | 1 | 5.80 |
| CHEMBL32301 | — | — | 1 | 5.52 |
| CHEMBL32940 | — | — | 1 | 5.36 |
| CHEMBL287256 | — | — | 1 | 5.03 |
| CHEMBL32248 | — | — | 1 | 5.03 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL33650 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL32301 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL32940 | — | IC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL287256 | — | IC50 | = | 9400.0 | nM | 5.03 |
| CHEMBL32248 | — | IC50 | = | 9300.0 | nM | 5.03 |