Assay Detail
Binding
CHEMBL814317
Review assay metadata, readout intent, target linkage, and publication context from the same page.
The inhibitory activity against thrombin (IIa)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Novel acylguanidine containing thrombin inhibitors with reduced basicity at the P1 moiety.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.82 | 7.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL114715 | INOGATRAN | 2.0 | 1 | 7.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL114715 | INOGATRAN | Ki | = | 15.0 | nM | 7.82 |