Assay Detail
Binding
CHEMBL814332
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Compound was evaluated for inhibition of Microbial tyramine oxidase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Fluorinated phenylcyclopropylamines. 1. Synthesis and effect of fluorine substitution at the cyclopropane ring on inhibition of microbial tyramine oxidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.83 | 7.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL500093 | — | — | 1 | 7.48 |
| CHEMBL51601 | — | — | 1 | 6.18 |
| CHEMBL903 | HYDRAZINECARBOXAMIDE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL500093 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL51601 | — | IC50 | = | 660.0 | nM | 6.18 |
| CHEMBL903 | HYDRAZINECARBOXAMIDE | IC50 | = | 6.7 | nM | - |