Assay Detail
Binding
CHEMBL814733
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Dissociation constant was determined from radioligand binding studies in human platelet membranes using Thromboxane A2 receptor radioligand [3H]-SQ 29,548.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Interphenylene phenyl oxazoles: novel, potent thromboxane receptor antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 8.86 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL31765 | — | — | 1 | 10.00 |
| CHEMBL170747 | — | — | 1 | 7.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL31765 | — | Kd | = | 0.1 | nM | 10.00 |
| CHEMBL170747 | — | Kd | = | 19.0 | nM | 7.72 |