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Assay Detail

CHEMBL814946

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards thrombin was determined
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Prothrombin (CHEMBL204)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery and development of the novel potent orally active thrombin inhibitor N-(9-hydroxy-9-fluorenecarboxy)prolyl trans-4-aminocyclohexylmethyl amide (L-372,460): coapplication of structure-based design and rapid multiple analogue synthesis on solid support.
Brady SF, Stauffer KJ, Lumma WC, Smith GM, Ramjit HG, Lewis SD, Lucas BJ, Gardell SJ, Lyle EA, Appleby SD, Cook JJ, Holahan MA, Stranieri MT, Lynch JJ, Lin JH, Chen IW, Vastag K, Naylor-Olsen AM, Vacca JP.
J Med Chem (1998) 41 : 401 -406
PubMed 9464370 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 8 8.75 10.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2062141 1 10.05
CHEMBL416795 1 10.00
CHEMBL364255 1 8.82
CHEMBL434417 1 8.60
CHEMBL131999 1 8.60
CHEMBL130119 1 8.52
CHEMBL125181 1 8.31
CHEMBL420689 1 7.12

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2062141 Ki = 0.09 nM 10.05
CHEMBL416795 Ki = 0.1 nM 10.00
CHEMBL364255 Ki = 1.5 nM 8.82
CHEMBL434417 Ki = 2.5 nM 8.60
CHEMBL131999 Ki = 2.5 nM 8.60
CHEMBL130119 Ki = 3.0 nM 8.52
CHEMBL125181 Ki = 4.9 nM 8.31
CHEMBL420689 Ki = 75.0 nM 7.12