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Assay Detail

CHEMBL815152

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards Trypsin.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Trypsin II (CHEMBL4472)
Type SINGLE PROTEIN
Organism Bos taurus

Publication

Design of benzamidine-type inhibitors of factor Xa.
Gabriel B, Stubbs MT, Bergner A, Hauptmann J, Bode W, Stürzebecher J, Moroder L.
J Med Chem (1998) 41 : 4240 -4250
PubMed 9784099 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.21 6.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL19902 DX-9065A 1 6.21

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL19902 DX-9065A Ki = 620.0 nM 6.21