Assay Detail
Binding
CHEMBL815360
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was tested for competitive inhibition with radioligand [3H]colchicine at colchicine site of mammalian tubulin
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Synthesis and biological properties of 1069C: a new synthetic antitumour agent with very low cross-resistance potential
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.12 | 6.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL418565 | — | — | 1 | 6.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL418565 | — | Ki | = | 750.0 | nM | 6.12 |